Atorvastatin

Administration

  • Type: Statins (HMG-CoA Reductase Inhibitor)
  • Dosage Forms:
  • Routes of Administration: PO
  • Common Trade Names: Lipitor

Adult Dosing

Hyperlipidemia

  • Moderate Intensity: 10-20 mg PO daily
  • High Intensity: 40-80 mg PO daily

Acute Coronary Syndrome

  • 80 mg PO (Single dose prior to PCI)

Pediatric Dosing

Special Populations

  • Pregnancy Rating: X
  • Lactation risk: Generally not recommended while breastfeeding
  • Renal Dosing
    • No adjustment
  • Hepatic Dosing
    • Contraindicated in patients with active liver disease

Contraindications

  • Allergy to class/drug

Adverse Reactions

Serious

  • Hepatotoxicity
  • Rhabdomyolysis

Common

  • Arthralgias
  • Dyspepsia
  • Nausea
  • UTI
  • Insomnia

Pharmacology

  • Half-life:
  • Metabolism:
  • Excretion:

Mechanism of Action

Comments

See Also

References